Research areas

  1. Published

    Thermal and acid denaturation of bovine lens a-crystallin

    Rasmussen, T., van de Weert, Marco, Jiskoot, W. & Kasimova, M. R., 2011, In: Proteins - Structure Function and Bioinformatics. 79, 6, p. 1747-1758

    Research output: Contribution to journalJournal articleResearchpeer-review

  2. Published

    Functionalization with ApoE-derived peptides enhances the interaction with brain capillary endothelial cells of nanoliposomes binding amyloid-beta peptide

    Re, F., Cambianica, I., Sesana, S., Salvati, E., Cagnotto, A., Salmona, M., Couraud, P., Moghimi, S. M., Masserini, M. & Sancini, G., 2011, In: Journal of Biotechnology. 156, 4, p. 341-346

    Research output: Contribution to journalJournal articleResearchpeer-review

  3. Published

    The spared nerve injury (SNI) model of induced mechanical allodynia in mice

    Richner, M., Bjerrum, Ole Jannik, Nykjær, A. & Vaegter, C. B., 18 Aug 2011, In: Journal of Visualized Experiments. 54, p. e3092

    Research output: Contribution to journalJournal articleResearchpeer-review

  4. Published

    Antistoffer produceret i bakterier

    Riise, E. S. & Skottrup, P. D., 2011, Bioteknologi - en temabog. Gasbjerg, P., Jensen, G. & Sørensen, A. (eds.). Aarhus: Systime Academic, p. 121-130 10 p.

    Research output: Chapter in Book/Report/Conference proceedingBook chapterEducation

  5. Published

    Acetylcholine binding protein as model of alpha4beta2 nicotinic acetylcholine receptors: Structural and functional characterization

    Rohde, L. A. H., 19 Dec 2011, København: Det Farmaceutiske Fakultet. 104 p.

    Research output: Book/ReportPh.D. thesisResearch

  6. Published

    Simulating kinetic parameters in transporter mediated permeability across Caco-2 cells. A case study of estrone-3-sulfate

    Rolsted, K., Rapin, N. P. J. & Steffansen, B., 2011, In: European Journal of Pharmaceutical Sciences. 44, 3, p. 218-226

    Research output: Contribution to journalJournal articleResearchpeer-review

  7. Published

    Hippocampal betaine/GABA transporter mRNA expression is not regulated by inflammation or dehydration post-status epilepticus

    Rowley, N. M., Smith, M. D., Lamb, J. G., Schousboe, Arne & White, H. S., 2011, In: Journal of Neurochemistry. 117, 1, p. 82-90

    Research output: Contribution to journalJournal articleResearchpeer-review

  8. Published

    Human phenotypically distinct TGFBI corneal dystrophies are linked to the stability of the fourth FAS1 domain of TGFBIp

    Runager, K., Basaiawmoit, R. V., Deva, T., Andreasen, M., Valnickova, Z., Sørensen, C. S., Karring, H., Thøgersen, I. B., Christiansen, G., Underhaug, J., Kristensen, T., Nielsen, N. C., Klintworth, G. K., Otzen, D. E. & Enghild, J. J., 18 Feb 2011, In: The Journal of Biological Chemistry. 286, 7, p. 4951-4958

    Research output: Contribution to journalJournal articleResearchpeer-review

  9. Published

    Computeren forudsiger lægemidlers omdannelse i leveren

    Rydberg, P. & Olsen, L., Dec 2011, In: Lægemiddelforskning. 2011, p. 44-46

    Research output: Contribution to journalJournal articleCommunication

  10. Published

    Do two different reaction mechanisms contribute to the hydroxylation of primary amines by cytochrome P450?

    Rydberg, P. & Olsen, L., Sep 2011, In: Journal of Chemical Theory and Computation. 7, 10, p. 3399-3404

    Research output: Contribution to journalJournal articleResearchpeer-review

  11. Published

    Evaluation of immunomodulating and anti-inflammatory effects of a herbal remedy based on rose hip powder (Rosa canina L.)

    Saaby, Lasse, 2011, København: Det Farmaceutiske Fakultet. 130 p.

    Research output: Book/ReportPh.D. thesisResearch

  12. Published

    Isolation of immunomodulatory triterpene acids from a standardized rose hip powder (Rosa canina L.)

    Saaby, Lasse, Jäger, A. K., Moesby, L., Hansen, E. W. & Christensen, Søren Brøgger, Feb 2011, In: Phytotherapy Research. 25, 2, p. 195-201

    Research output: Contribution to journalJournal articleResearchpeer-review

  13. Published

    Ubiquitous plant compounds disturb cell-based assays

    Saaby, Lasse & Jäger, A. K., 1 Sep 2011, In: Journal of Ethnopharmacology. 137, 1, p. 942-943

    Research output: Contribution to journalComment/debateResearchpeer-review

  14. Published

    Combined MUC1-specific nanobody-tagged PEG-polyethylenimine polyplex targeting and transcriptional targeting of tBid transgene for directed killing of MUC1 over-expressing tumour cells

    Sadeqzadeh, E., Rahbarizadeh, F., Ahmadvand, D., Rasaee, M. J., Parhamifar, L. & Moghimi, S. M., 2011, In: Journal of Controlled Release. 156, 1, p. 85-91

    Research output: Contribution to journalJournal articleResearchpeer-review

  15. Published

    New insights into the GABAA receptor structure and orthosteric ligand binding: Receptor modeling guided by experimental data

    Sander, T., Frølund, Bente, Bruun, A. T., Ivanov, I., McCammon, J. A. & Balle, T., May 2011, In: Proteins: Structure, Function, and Bioinformatics. 79, 5, p. 1458-1477

    Research output: Contribution to journalJournal articleResearchpeer-review

  16. Published

    Neuron-glia interactions in glutamatergic neurotransmission: roles of oxidative and glycolytic adenosine triphosphate as energy source

    Schousboe, Arne, Sickmann, H. M., Bak, Lasse Kristoffer, Schousboe, I., Jajo, F. S., Faek, S. A. A. & Waagepetersen, Helle S., 1 Dec 2011, In: Journal of Neuroscience Research. 89, 12, p. 1926-34 9 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  17. Published

    GABA transport inhibitors and seizure protection: the past and future

    Schousboe, Arne, Madsen, K. K. & White, S., 2011, In: Future Medicinal Chemistry. 3, 2, p. 183-187 5 p.

    Research output: Contribution to journalReviewResearchpeer-review

  18. Published

    Perceived pain communication among Lithuanian cancer patients

    Sciupokas, A., Liubarskiene, Z., Samsanaviciene, J. & Jacobsen, Ramune, 2011.

    Research output: Contribution to conferenceConference abstract for conferenceResearch

  19. Published

    Characterization of capsaicin induced responses in mice vas deferens: evidence of CGRP uptake

    Sheykhzade, Majid, Gupta, S., Sørensen, T., Sørensen, O. A., Koch, H., Boonen, H. C. M., Back, O. & Fjalland, B., 2011, In: European Journal of Pharmacology. 667, 1-3, p. 375-382

    Research output: Contribution to journalJournal articleResearchpeer-review

  20. Published

    Diagnostic evaluation of a nanobody with picomolar affinity toward the protease RgpB from Porphyromonas gingivalis

    Skottrup, P. D., Leonard, P., Kaczmarek, J., Veillard, F., Johannes Enghild, J., O'Kennedy, R., Sroka, A., Clausen, Rasmus Prætorius, Potempa, J. & Riise, E. S., 2011, In: Analytical Biochemistry. 415, 2, p. 158-167

    Research output: Contribution to journalJournal articleResearchpeer-review

  21. Published

    Nanobodies fra kameler - En ny klasse antistoffer til diagnostik og behandling

    Skottrup, P. D., Clausen, Rasmus Prætorius & Riise, E., Dec 2011, In: Lægemiddelforskning. 2011, p. 4-6

    Research output: Contribution to journalJournal articleCommunication

  22. Published

    The cysteine protease RgpB as a biomarker for the periodonto-pathogen Porphyromonas gingivalis: Nanobody selection and assay development

    Skottrup, P. D., Leonard, P., Kaczmarek, J., Veillard, F., Johannes Enghild, J., O'Kennedy, R., Sroka, A., Clausen, Rasmus Prætorius, Potempa, J. & Riise, E. S., 2011.

    Research output: Contribution to conferencePosterResearch

  23. Published

    Myocardial ischemia-reperfusion induces upregulation of contractile endothelin ETB receptor in rat coronary arteries

    Skovsted, G. F., Sheykhzade, Majid, Trautner, S. & Edvinsson, L., 2011, In: pA2 online. 9, 1, 1 p.

    Research output: Contribution to journalConference abstract in journalResearchpeer-review

  24. Published

    The calcium-sensing receptor and calcimimetics in blood pressure modulation

    Smajilovic, S., Yano, S., Jabbari, R. & Tfelt-Hansen, J., Oct 2011, In: British Journal of Pharmacology. 164, 3, p. 884-893

    Research output: Contribution to journalReviewResearchpeer-review

  25. Published

    Expression and beta-glucan binding properties of Scots pine (Pinus sylvestris L.) antimicrobial protein (Sp-AMP)

    Sooriyaarachchi, S., Jaber, E., Covarrubias, A. S., Ubhayasekera, W., Asiegbu, F. O. & Mowbray, S. L., 17 May 2011, In: Plant Molecular Biology. 77, 1-2, p. 33-45

    Research output: Contribution to journalJournal articleResearchpeer-review

  26. Published

    Effects of Teucrium polium spp. capitatum flavonoids on the lipid and carbohydrate metabolism in rats

    Stefkov, G., Kulevanova, S., Miova, B., Dinevska-Kjovkarovska, S., Mølgaard, Per, Jäger, A. K. & Josefsen, K., 1 Sep 2011, In: Pharmaceutical Biology. 49, 9, p. 885-892

    Research output: Contribution to journalJournal articleResearchpeer-review

  27. Published

    Calu-3 cells grown under AIC and LCC conditions: implications for dipeptide uptake and transepithelial transport of substances

    Stentebjerg-Andersen, A., Notlevesen, I. V., Larsen, Birger Brodin & Nielsen, C. U., 2011, In: European Journal of Pharmaceutics and Biopharmaceutics. 78, 1, p. 19-26

    Research output: Contribution to journalJournal articleResearchpeer-review

  28. Published

    Structural basis of slow activation gating in the cardiac IKs channel complex

    Strutz-Seebohm, N., Pusch, M., Wolf, S., Stoll, R., Tapken, D., Gerwert, K., Attali, B. & Seebohm, G., 2011, In: Cellular Physiology and Biochemistry. 27, 5, p. 443-452

    Research output: Contribution to journalJournal articleResearchpeer-review

  29. Published

    Electrophilic organic selenium reagents: protonated seleninic acids as precursors for unsymmetrical aromatic selenides

    Stuhr-Hansen, N., Sølling, Theis Ivan & Henriksen, L., 8 Apr 2011, In: Tetrahedron. 67, 14, p. 2633-2643

    Research output: Contribution to journalJournal articleResearchpeer-review

  30. Published

    Environmental risk assessment of three selective serotonin reuptake inhibitors in the aquatic environment: A case study including a cocktail scenario

    Styrishave, Bjarne, Halling-Sørensen, B. & Ingerslev, F., 2011, In: Environmental Toxicology and Chemistry. 30, 1, p. 254-261

    Research output: Contribution to journalJournal articleResearchpeer-review

  31. Published

    Evolution and applications of plant pathway resources and databases

    Sucaet, Y. & Deva, T., Sep 2011, In: Briefings in Bioinformatics. 12, 5, p. 530-544

    Research output: Contribution to journalJournal articleResearchpeer-review

  32. Published

    Antifungal metabolites from fungal endophytes of Pinus strobus

    Sumarah, M. W., Kesting, J. R., Sørensen, D. & Miller, J. D., 1 Oct 2011, In: Phytochemistry. 72, 14-15, p. 1833-1837

    Research output: Contribution to journalJournal articleResearchpeer-review

  33. Published

    Kv7 positive modulators reduce detrusor over-activity and increase bladder capacity in rats

    Svaloe, J., Hansen, H. H., Rønn, L. C. B., Sheykhzade, Majid, Munro, G. J. & Rode, F., 2011, In: Basic & Clinical Pharmacology & Toxicology. 110, 2, p. 145-153

    Research output: Contribution to journalJournal articleResearchpeer-review

  34. Published

    A new phenylalanine derivative acts as an antagonist at the AMPA receptor GluA2 and introduces partial domain closure: Synthesis, resolution, pharmacology, and crystal structure

    Szymanska, E., Frydenvang, Karla Andrea, Contreras-Sanz, A., Pickering, Darryl S, Frola, E., Serafimoska, Z., Nielsen, Birgitte, Kastrup, Jette Sandholm Jensen & Johansen, Tommy Nørskov, 4 Oct 2011, In: Journal of Medicinal Chemistry. 54, 20, p. 7289-7298

    Research output: Contribution to journalJournal articleResearchpeer-review

  35. Published

    Medicingennemgang-en ydelse i sundhedssektoren? Notat fra debatmøde for beslutningstagere og interesseorganisationer i sundhedssektoren

    projektgruppen for Medisam-projektet, P. F. M., 2011, Medisam. København: Det Farmaceutiske Fakultet, 8 p.

    Research output: Chapter in Book/Report/Conference proceedingReport chapterResearch

  36. Published

    Medisam- en samarbejdsmodel til medicingennemgang og medicinafstemning mellem patienter, læger,apotek: Afsluttende rapport

    Projektgruppen for Medisam projektet, P. F. M. P., 2011, København: Det Farmaceutiske Fakultet. 8 p.

    Research output: Book/ReportReportResearch

  37. Published

    Studies of monoamine transporters: Phosphorylation of the serotonin transporter and interactions of antidepressants with the serotonin and norepinephrine transporters

    Sørensen, L., May 2011, København: Det Farmaceutiske Fakultet. 174 p.

    Research output: Book/ReportPh.D. thesisResearch

  38. Published

    Amaryllidaceae alkaloids from the Australasian tribe Calostemmateae with acetylcholinesterase inhibitory activity

    Søvsø Jensen, B., Christensen, Søren Brøgger, Jäger, A. K. & Rønsted, Nina, Apr 2011, In: Biochemical Systematics and Ecology. 39, 2, p. 153-155

    Research output: Contribution to journalJournal articleResearchpeer-review

  39. Published

    In silico predictions of hERG channel blockers in drug discovery: from ligand-based and target-based approaches to systems chemical biology

    Taboureau, O. & Jørgensen, Flemming Steen, Jun 2011, In: Combinatorial Chemistry & High Throughput Screening. 14, 5, p. 375-387

    Research output: Contribution to journalJournal articleResearchpeer-review

  40. Published

    The quest for targeted delivery in colon cancer: mucoadhesive valdecoxib microspheres

    Thakral, N. K., Ray, A. R., Bar-Shalom, Daniel, Eriksson, A. H. & Majumdar, D. K., 2011, In: International Journal of Nanomedicine. 6, p. 1057-1068

    Research output: Contribution to journalJournal articleResearchpeer-review

  41. Published

    Pharmacological and physiological studies of the calcium-sensing receptor

    Thomsen, A. R. B., Nov 2011, København: Det Farmaceutiske Fakultet. 89 p.

    Research output: Book/ReportPh.D. thesisResearch

  42. Published

    The tandem chain extension aldol reaction used for synthesis of ketomethylene tripeptidomimetics targeting hPEPT1

    Thorn, K., Nielsen, C. U., Jakobsen, P., Steffansen, B., Zercher, C. K. & Begtrup, M., Aug 2011, In: Bioorganic & Medicinal Chemistry Letters. 21, 15, p. 4597-4601

    Research output: Contribution to journalJournal articleResearchpeer-review

  43. Published

    Analysis of secondary plant metabolites by indirect desorption electrospray ionization imaging mas spectrometry

    Thunig, U. J. C., Hansen, S. H. & Janfelt, Christian, 2011, In: Analytical Chemistry. 83, p. 3256-3259

    Research output: Contribution to journalLetterResearchpeer-review

  44. Published

    Perspective on water of crystallization affecting the functionality of pharmaceuticals

    Tian, F. & Rantanen, Jukka, 2011, In: Food Biophysics. 6, 2, p. 250-258

    Research output: Contribution to journalJournal articleResearchpeer-review

  45. Published

    Preparing students for industrial quality control of medicines while keeping a problem-based and research-oriented learning environment

    Timm, M., 2011, Improving university science teaching and learning: Pedagogical projects 2010. 1 ed. Copenhagen, Denmark, Vol. 3/1. p. 189-207 19 p.

    Research output: Chapter in Book/Report/Conference proceedingBook chapterEducation

  46. Published

    Brute-force pharmacophore assessment and scoring with Open3DQSAR

    Tosco, P. & Balle, T., 2011, In: Journal of Cheminformatics. 3, Suppl 1, p. 22

    Research output: Contribution to journalConference abstract in journalResearchpeer-review

  47. Published

    Open3DALIGN: an open-source software aimed at unsupervised ligand alignment

    Tosco, P., Balle, T. & Shiri, F., 27 Jul 2011, In: Journal of Computer - Aided Molecular Design. 25, 8, p. 777-783

    Research output: Contribution to journalJournal articleResearchpeer-review

  48. Published

    Open3DGRID: An open-source software aimed at high-throughput generation of molecular interaction fields (MIFs)

    Tosco, P. & Balle, T., 2011

    Research output: Non-textual formComputer programmeResearch

  49. Published

    Open3DQSAR: a new open-source software aimed at high-throughput chemometric analysis of molecular interaction fields

    Tosco, P. & Balle, T., 2011, In: Journal of Molecular Modeling. 17, 1, p. 201-208

    Research output: Contribution to journalJournal articleResearchpeer-review

  50. Published

    Open3DQSAR: An open-source software aimed at high-throughput chemometric analysis of molecular interaction fields

    Tosco, P. & Balle, T., 2011

    Research output: Non-textual formComputer programmeResearch

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