Research areas

  1. Published

    Neuroprotective and neurochemical properties of mint extracts

    López, V., Martín, S., Gómez-Serranillos, M. P., Carretero, M. E., Jäger, A. K. & Calvo, M. I., 2010, In: Phytotherapy Research. 24, 6, p. 869-874

    Research output: Contribution to journalJournal articleResearchpeer-review

  2. Published

    Synthesis of imidazole-4(5)-acetic acid analogues: for characterizing the ionotropic GABA receptors

    Madsen, C., 2010, København: Det Farmaceutiske Fakultet. 186 p.

    Research output: Book/ReportPh.D. thesisResearch

  3. Published

    Investigation of the interaction between modified ISCOMs and stratum corneum lipid model systems

    Madsen, H. B., Arboe-Andersen, H. M., Rozlosnik, N., Madsen, F., Ifversen, P., Kasimova, M. R. & Nielsen, Hanne Mørck, 2010, In: Biochimica et Biophysica Acta - Biomembranes. 1798, p. 1779-1789

    Research output: Contribution to journalJournal articleResearchpeer-review

  4. Published

    Penetration and interaction of ISCOM nanoparticles with the skin

    Madsen, H. B., 2010, København: Museum Tusculanum. 73 p.

    Research output: Book/ReportPh.D. thesisResearch

  5. Published

    Neuronal and non-neuronal GABA transporters as targets for antiepileptic drugs

    Madsen, K. K., White, H. S. & Schousboe, Arne, 2010, In: Pharmacology & Therapeutics. 125, 3, p. 394-401

    Research output: Contribution to journalJournal articleResearchpeer-review

  6. Published

    Ribavirin dosage in patients with HCV genotypes 2 and 3 who completed short therapy with peg-interferon alpha-2b and ribavirin

    Mangia, A., Dalgard, O., Minerva, N., Verbaan, H., Bacca, D., Larsen, H. R., Copetti, M., Caretta, V., Piazzollla, V., Cozzolongo, R., Mottola, L. & Andriulli, A., 1 Jun 2010, In: Alimentary Pharmacology and Therapeutics. 31, 12, p. 1346-53 7 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  7. Published

    Building the quality into pellet manufacturing environment - Feasibility study and validation of an in-line quantitative near infrared (NIR) method

    Mantanus, J., Ziémons, E., Rozet, E., Streel, B., Klinkenberg, R., Evrard, B., Rantanen, Jukka & Hubert, P., 2010, In: Talanta: The International Journal of Pure and Applied Analytical Chemistry. 83, 2, p. 305-311

    Research output: Contribution to journalJournal articleResearch

  8. Published

    Using a phylogenetic approach to selection of target plants in drug discovery of acetylcholinesterase inhibiting alkaloids in Amaryllidaceae tribe Galantheae

    Mellergaard Larsen, M., Adsersen, A., Davis, A. P., Lledó, M. D., Jäger, A. K. & Rønsted, Nina, Oct 2010, In: Biochemical Systematics and Ecology. 38, 5, p. 1026-1034

    Research output: Contribution to journalJournal articleResearchpeer-review

  9. Published

    Regional differences in reporting patterns for adverse drug reactions: a retrospective analysis of reports from 2000 to 2009 in Vigibase

    Melskens, L., Petersen, P. S. & Aagaard, L., 2010, In: Drug Safety. 33, 10, p. 902-903

    Research output: Contribution to journalConference abstract in journalResearch

  10. Published

    Complement activation cascade triggered by PEG-PL engineered nanomedicines and carbon nanotubes: The challanges ahead

    Moghimi, S. M., Andersen, A. J., Hashemi, S. H., Lettiero, B., Ahmadvand, D., Hunter, A. C., Andresen, T. L., Hamad, I. & Szebeni, J., 2010, In: Journal of Controlled Release. 146, 2, p. 175-181

    Research output: Contribution to journalJournal articleResearchpeer-review

  11. Published

    Complement monitoring of carbon nanotubes

    Moghimi, S. M. & Hunter, A. C., 2010, In: Nature Nanotechnology. 5, p. 382-382

    Research output: Contribution to journalComment/debateResearchpeer-review

  12. Published

    Nanomedicine and nanotoxicology at Pharma-Copenhagen University

    Moghimi, S. M., Hashemi, S. H., Larsen, A. K., Parhamifar, L., Ahmadvand, D., Andersen, A. J., Wu, L. & Lettiero, B., 2010, In: European Journal of Nanomedicine. 3, 1, p. 41-43

    Research output: Contribution to journalJournal articleResearchpeer-review

  13. Published

    Extensive small-angle X-ray scattering studies of blood coagulation factor VIIa reveal interdomain flexibility

    Mosbæk, C. R., Nolan, D., Persson, E., Svergun, D. I., Bukrinsky, J. T. & Vestergaard, Bente, 2010, In: Biochemistry. 49, 45, p. 9739-9745

    Research output: Contribution to journalJournal articleResearchpeer-review

  14. Published

    Small angle X-ray scattering studies of blood coagulation factor VII and antibodies at high concentration

    Mosbæk, C. R., 12 Oct 2010, København: Det Farmaceutiske Fakultet. 141 p.

    Research output: Book/ReportPh.D. thesisResearch

  15. Published

    Quinazolin-4-one derivatives: A novel class of noncompetitive NR2C/D subunit-selective N-methyl-D-aspartate receptor antagonists

    Mosley, C. A., Acker, T. M., Hansen, K. B., Mullasseril, P., Andersen, K. T., Le, P., Vellano, K. M., Bräuner, Hans, Liotta, D. C. & Traynelis, S. F., 2010, In: Journal of Medicinal Chemistry. 53, 15, p. 5476-5490

    Research output: Contribution to journalJournal articleResearchpeer-review

  16. Published

    Production and nutritional aspects of human milk fat substitutes

    Mu, Huiling, 2010, In: Lipid Technology. 22, 6, p. 126-129

    Research output: Contribution to journalJournal articleResearchpeer-review

  17. Published

    "Patients don't lie"; a view on adherence in asthma

    Møldrup, C., Stein, J. & Søndergaard, B., 2010, In: Pharmacy World and Science. 32, 6, p. 795-798

    Research output: Contribution to journalJournal articleResearchpeer-review

  18. Published

    Effect of the cannabinoid receptor-1 antagonist rimonabant on lipolysis in rats

    Mølhøj, S., Hansen, Harald S., Schweiger, M., Zimmermann, R., Johansen, T. & Malmlöf, K., 2010, In: European Journal of Pharmacology. 646, 1-3, p. 38-45

    Research output: Contribution to journalJournal articleResearchpeer-review

  19. Published

    Stability, liposome interaction, and in vivo pharmacology of ghrelin in liposomal suspensions

    Møller, E. H., Holst, Birgitte, Nielsen, L. H., Pedersen, P. S. & Østergaard, Jesper, 2010, In: Internation Journal of Pharmaceutics. 390, 1, p. 13-18

    Research output: Contribution to journalJournal articleResearchpeer-review

  20. Published

    Novel 4-(piperidin-4-yl)-1-hydroxypyrazoles as gamma-aminobutyric acidA receptor ligands: synthesis, pharmacology, and structure-activity relationships

    Møller, H. A., Sander, T., Kristensen, Jesper Langgaard, Nielsen, Birgitte, Krall, J., Bergmann, M. L., Christiansen, B., Balle, T., Jensen, Anders A. & Frølund, Bente, 2010, In: Journal of Medicinal Chemistry. 53, 8, p. 3417-3421

    Research output: Contribution to journalJournal articleResearchpeer-review

  21. Published

    Insights into the ultrastructure of human intestinal fluids in the fed state by electron microscopy analysis

    Mullertz, Anette , Fatouros, D., Smith, J. R., Vertzoni, M. & Rappas, C., Nov 2010.

    Research output: Contribution to conferencePosterResearch

  22. Published

    Effect of GTP-cyclohydrolase deficiency in the HPH-1mouse on acute and inflammatory pain

    Nasser, A., Bjerrum, Ole Jannik & Heegaard, Anne-Marie, 2010.

    Research output: Contribution to conferenceConference abstract for conferenceCommunication

  23. Published

    Genetik kan forudsige følsomhed for smerte

    Nasser, A., Bjerrum, Ole Jannik, Heegaard, Anne-Marie & Møller, L. B., 2010, In: Lægemiddelforskning. 2010, p. 34-36

    Research output: Contribution to journalJournal articleResearch

  24. Published

    The GTP-cyclohydrolase deficient mouse shows reduced acute pain perception

    Nasser, A., Bjerrum, Ole Jannik, Heegaard, Anne-Marie & Møller, L. B., 2010.

    Research output: Contribution to conferencePosterCommunication

  25. Published

    Serotonin transporter affinity of (-)-loliolide, a monoterpene lactone from Mondia whitei

    Neergaard, J. S., Rasmussen, H. B., Stafford, G. I., van Staden, J. & Jäger, A. K., 2010, In: South African Journal of Botany. 76, 3, p. 593-596

    Research output: Contribution to journalJournal articleResearchpeer-review

  26. Published

    Neuropathic pain: sortilin is involved in the down-regulation of KCC2

    Neustrup, S., P., M., Bjerregaard, C. V., Nykjær, A. & Bjerrum, Ole Jannik, 2010.

    Research output: Contribution to conferencePosterCommunication

  27. Published

    Absorptive transporters

    Nielsen, C. U., Steffansen, B. & Larsen, Birger Brodin, 2010, Molecular biopharmaceutics: Aspects of drug characterisation, drug delivery and dosage from evaluation. Steffansen, B., Brodin, B. & Uhd Nielsen, C. (eds.). London: Pharmaceutical Press, p. 193-211 (ULLA Pharmacy Series).

    Research output: Chapter in Book/Report/Conference proceedingBook chapterResearchpeer-review

  28. Published

    Carrier-mediated transport kinetics

    Nielsen, C. U., Steffansen, B. & Larsen, Birger Brodin, 2010, Molecular biopharmaceutics: Aspects of drug characterisation, drug delivery and dosage form evaluation. Pharmaceutical Press, p. 153-173

    Research output: Chapter in Book/Report/Conference proceedingBook chapterResearchpeer-review

  29. Published

    Efflux transporters

    Nielsen, C. U., Larsen, Birger Brodin & Steffansen, B., 2010, Molecular biopharmaceutics: Aspects of drug characterisation, drug delivery and dosage form evaluation. Steffansen, B., Brodin, B. & Uhd Nielsen, C. (eds.). Pharmaceutical Press, p. 213-22

    Research output: Chapter in Book/Report/Conference proceedingBook chapterResearchpeer-review

  30. Published

    GABA transport across the basolateral membrane of intestinal cells

    Nielsen, C. U., Carstensen, M. & Larsen, Birger Brodin, 2010. 1 p.

    Research output: Contribution to conferenceConference abstract for conferenceResearchpeer-review

  31. Published

    Amination of aryl iodides using a fluorous-tagged ammonia equivalent

    Nielsen, S. D., Smith, G., Begtrup, M. & Kristensen, Jesper Langgaard, 2010, In: European Journal of Organic Chemistry. 2010, 19, p. 3704-3710

    Research output: Contribution to journalJournal articleResearchpeer-review

  32. Published

    Synthesis and application of a new fluorous-tagged ammonia equivalent

    Nielsen, S. D., Smith, G., Begtrup, M. & Kristensen, Jesper Langgaard, 2010, In: Chemistry: A European Journal. 16, 15, p. 4557-4566

    Research output: Contribution to journalJournal articleResearchpeer-review

  33. Published

    Investigation of the mnemonic deficits in the sub-chronic PCP model of schizophrenia

    Nielsen, T. D., 2010, København: Museum Tusculanum. 73 p.

    Research output: Book/ReportPh.D. thesisResearch

  34. Published

    Positive modulation of alpha-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid (AMPA) receptors reverses subcronic PCP-induced deficits in the novel object recognition task in rats

    Nielsen, T. D., Larsen, D. B., Hansen, S. L., Grayson, B., Neill, J. C. & Plath, N., 11 Feb 2010, In: Behavioural Brain Research. 207, 1, p. 144-150 7 p.

    Research output: Contribution to journalJournal articleResearch

  35. Published

    Application of Q2MM to stereoselective reactions

    Nilsson Lill, S. O., Forbes, A., Donoghue, P., Verdolino, V., Wiest, O., Rydberg, P. & Norrby, P., Sep 2010, In: Current Organic Chemistry. 14, 15, p. 1629-1645

    Research output: Contribution to journalReviewResearchpeer-review

  36. Published

    A synthetic mycobacterial monomycoloyl glycerol analogue stabilizes DDA liposomes

    Nordly, P. J., Pedersen, E. A., Khiljii, T. S., Agger, E. M., Jørgensen, Lene, Nielsen, Hanne Mørck, Korsholm, K. S., Franzyk, Henrik & Foged, Camilla, 2010, In: CRS Newsletter. 27, 2, p. 12 14 p.

    Research output: Contribution to journalJournal articleResearch

  37. Published

    Formulation of vaccine adjuvants: modulating the adjuvant activity of DDA/TDB liposomes with immunopotentiators

    Nordly, P. J., 2010, København: Det Farmaceutiske Fakultet.

    Research output: Book/ReportPh.D. thesisResearch

  38. Published

    Characterization of nanofilm spray products by mass spectrometry

    Nørgaard, A. W., Wolkoff, P. & Lauritsen, F. R., 2010, In: Chemosphere. 80, p. 1377-1386

    Research output: Contribution to journalJournal articleResearchpeer-review

  39. Published

    Real-time monitoring of the progerss of polymerization reactions directly on surfaces at open atmosphere by ambient mass spectrometry

    Nørgaard, A. W., Vaz, B. G., Lauritsen, F. R. & Eberlin, M. N., 2010, In: Rapid Communications in Mass Spectrometry. 24, p. 3441-3446

    Research output: Contribution to journalJournal articleResearchpeer-review

  40. Published

    From consumerism to active dependence: patterns of medicines use and treatment decisions among patients with atopic dermatitis

    Nørreslet, M., Bissell, P. & Traulsen, Janine Marie, 2010, In: Health. 14, 1, p. 91-106

    Research output: Contribution to journalJournal articleResearchpeer-review

  41. Published

    A pharmacokinetic and pharmacodynamic study of oral oxycodone in a human experimental pain model of hyperalgesia

    Olesen, A. E., Upton, R., Staahl, C., Christrup, Lona Louring, Arendt-Nielsen, L. & Drewes, A. M., 2010, In: Clinical Pharmacokinetics. 49, 12, p. 817-827

    Research output: Contribution to journalJournal articleResearchpeer-review

  42. Published

    Antimicrobial, hemolytic, and cytotoxic activities of ß-peptoid-peptide hybrid oligomers: Improved properties compared to natural AMPs

    Olsen, Christian Adam, Ziegler, H. L., Nielsen, Hanne Mørck, Frimodt-Møller, N., Jaroszewski, J. W. & Franzyk, Henrik, 2010, In: ChemBioChem. 11, 10, p. 1356-1360

    Research output: Contribution to journalJournal articleResearchpeer-review

  43. Published

    Peptoid-Peptide hybrid backbone architectures

    Olsen, Christian Adam, 25 Jan 2010, In: ChemBioChem. 11, 2, p. 152-160

    Research output: Contribution to journalJournal articleResearchpeer-review

  44. Published

    A quantitative structure-activity relationship for translocation of tripeptides via the human proton-coupled peptide transporter, hPEPT1 (SLC15A1)

    Omkvist, D. H., Larsen, S. B., Nielsen, C. U., Steffansen, B., Olsen, L., Jørgensen, Flemming Steen & Larsen, Birger Brodin, 2010, In: The AAPS Journal. 12, 3, p. 385-396

    Research output: Contribution to journalJournal articleResearchpeer-review

  45. Published

    Ibuprofen is a non-competitive inhibitor of the peptide transporter hPEPT1 (SLC15A1): possible interactions between hPEPT1 substrates and ibuprofen

    Omkvist, D. H., Larsen, Birger Brodin & Nielsen, C. U., 2010, In: British Journal of Pharmacology. 161, 8, p. 1793-1805

    Research output: Contribution to journalJournal articleResearchpeer-review

  46. Published

    Ibuprofen is an inhibitor of hPEPT1: Implications for drug-drug interactions at the level of drug absorption

    Omkvist, D. H., Larsen, Birger Brodin & Nielsen, C. U., 2010.

    Research output: Contribution to conferencePosterResearch

  47. Published

    Development of solid-phase aziridine chemistries: Piperazine scaffolds and unnatural amino acid building blocks

    Ottesen, L. K., 2010, København: Det Farmaceutiske Fakultet. 139 p.

    Research output: Book/ReportPh.D. thesisResearch

  48. Published

    Ring opening of a resin-bound chiral aziridine with phenol nucleophiles

    Ottesen, L. K., Jaroszewski, J. W. & Franzyk, Henrik, 2010, In: Journal of Organic Chemistry. 75, 15, p. 4983-4991

    Research output: Contribution to journalJournal articleResearchpeer-review

  49. Published

    Gold-embedded photosensitive liposomes for drug delivery: Triggering mechanism and intracellular release

    Paasonen, L., Sipilä, T., Subrizi, A., Laurinmäki, P., Butcher, S. J., Rappolt, M., Yaghmur, Anan, Urtti, A. & Yliperttula, M., 2010, In: Journal of Controlled Release. 147, p. 136-143

    Research output: Contribution to journalJournal articleResearchpeer-review

  50. Published

    Polycation cytotoxicity: a delicate matter for nucleic acid therapy - focus on polyethylenimine

    Parhamifar, L., Larsen, A. K., Hunter, A. C., Andresen, T. L. & Moghimi, S. M., 2010, In: Soft Matter. 6, p. 4001-4009

    Research output: Contribution to journalJournal articleResearchpeer-review

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